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1Chen Zhifeng, Zhang Hao, Liu Shien, Xie Yiqian, Jiang Hao, Lu Wenchao, Xu Heng, Yue Liyan, Zhang Yuanyuan, Ding Hong, Zheng Mingyue, Yu Kunqian, Chen Kaixian, Jiang Hualiang, Luo Cheng.
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay, Med. Chem. Commun., 2017