ChemSpider 2D Image | Tabimorelin | C68H84N8O10

Tabimorelin

  • Molecular FormulaC68H84N8O10
  • Average mass1173.442 Da
  • Monoisotopic mass1172.630981 Da
  • ChemSpider ID10154034
  • Double-bond stereo - Double-bond stereo


More details:






Validated by Experts, Validated by Users, Non-Validated, Removed by Users

(2E)-2-Butendisäure --N-[(2E)-5-amino-5-methyl-2-hexenoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamid (1:2) [German] [ACD/IUPAC Name]
193079-69-5 [RN]
Acide (2E)-2-butènedioïque - N-[(2E)-5-amino-5-méthyl-2-hexenoyl]-N-méthyl-3-(2-naphtyl)-D-alanyl-N,Nα-diméthyl-D-phénylalaninamide (1:2) [French] [ACD/IUPAC Name]
D-Phenylalaninamide, N-[(2E)-5-amino-5-methyl-1-oxo-2-hexen-1-yl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-dimethyl-, (2E)-2-butenedioate (2:1) [ACD/Index Name]
N-[(2E)-5-Amino-5-methyl-2-hexenoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-2-butenedioate (2:1) [ACD/IUPAC Name]
N-[(2E)-5-Amino-5-methylhex-2-enoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-but-2-enedioate (2:1)
Tabimorelin [INN] [Wiki]
[242143-80-2] [RN]
242143-80-2 [RN]
NN 703
More...
  • Experimental Physico-chemical Properties
    • Experimental Solubility:

      Soluble to 10 mM in water and to 100 mM in DMSO Tocris Bioscience 2308
      Soluble to 10 mM in water with gentle warming and to 100 mM in DMSO Tocris Bioscience 2308
  • Miscellaneous
    • Bio Activity:

      7-TM Receptors Tocris Bioscience 2308
      Ghrelin Receptors Tocris Bioscience 2308
      Peptide Receptors Tocris Bioscience 2308
      Potent, orally active ghrelin receptor (GHS-R1a) agonist (Ki = 50 nM at human recombinant GHS-R1a). Stimulates GH release from rat pituitary cells with an EC50 value of 2.7 nM. Induces hyperphagia and adiposity in lean rats, but not in leptin signaling-deficient ZDF rats. Tocris Bioscience 2308
      Potent, orally active ghrelin receptor (GHS-R1a) agonist (Ki = 50 nM at human recombinant GHS-R1a). Stimulates GH release from rat pituitary cells with an EC50 value of 2.7 nM. Induces hyperphagia and adiposity in lean rats, but not in leptin signaling-deficient ZDF rats. Tocris Bioscience 2308
      Potent, orally active ghrelin receptor agonist Tocris Bioscience 2308

Predicted data is generated using the ACD/Labs Percepta Platform - PhysChem Module, version: 14.00

No predicted properties have been calculated for this compound.

Click to predict properties on the Chemicalize site






Advertisement