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- Potential atypical antipsychotics: synthesis, binding affinity and SAR of new heterocyclic bioisosteric butyrophenone analogues as multitarget ligands. María Barceló, Enrique Raviña, María J. Varela, José Brea, María I. Loza, Christian F. Masaguer
, Med. Chem. Commun.
, 2011
, 2
, 1194
- Synthesis and evaluation of amide, sulfonamide and urea – benzisoxazole derivatives as potential atypical antipsychotics. Yin Chen, Yu Lan, Xudong Cao, Xiangqing Xu, Juecheng Zhang, Minquan Yu, Xin Liu, Bi-Feng Liu, Guisen Zhang
, Med. Chem. Commun.
, 2015
, 6
, 831
- Discovery of 4-benzoylpiperidine and 3-(piperidin-4-yl)benzo[d]isoxazole derivatives as potential and selective GlyT1 inhibitors. Yang Liu, Lin Guo, Hongliang Duan, Liming Zhang, Neng Jiang, Xuechu Zhen, Jianhua Shen
, RSC Adv.
, 2015
, 5
, 40964
- High-throughput identification of G protein-coupled receptor modulators through affinity mass spectrometry screening. Shanshan Qin, Mengmeng Meng, Dehua Yang, Wenwen Bai, Yan Lu, Yao Peng, Gaojie Song, Yiran Wu, Qingtong Zhou, Suwen Zhao, Xiping Huang, John D. McCorvy, Xiaoqing Cai, Antao Dai, Bryan L. Roth, Michael A. Hanson, Zhi-Jie Liu, Ming-Wei Wang, Raymond C. Stevens, Wenqing Shui
, Chem. Sci.
, 2018
, 9
, 3192
- Machine learning vs. field 3D-QSAR models for serotonin 2A receptor psychoactive substances identification. Giuseppe Floresta, Vincenzo Abbate
, RSC Adv.
, 2021
, 11
, 14587
- Pharmacophore-based tailoring of biphenyl amide derivatives as selective 5-hydroxytryptamine 2B receptor antagonists. Moustafa T. Gabr, Mohammed S. Abdel-Raziq
, Med. Chem. Commun.
, 2018
, 9
, 1069
- Development of selective agents targeting serotonin 5HT1A receptors with subnanomolar activities based on a coumarin core. K. Ostrowska, D. Grzeszczuk, M. Głuch-Lutwin, A. Gryboś, A. Siwek, Ł. Dobrzycki, B. Trzaskowski
, Med. Chem. Commun.
, 2017
, 8
, 1690
- Search for a 5-CT alternative. In vitro and in vivo evaluation of novel pharmacological tools: 3-(1-alkyl-1H-imidazol-5-yl)-1H-indole-5-carboxamides, low-basicity 5-HT7 receptor agonists. Gniewomir Latacz, Adam S. Hogendorf, Agata Hogendorf, Annamaria Lubelska, Joanna M. Wierońska, Monika Woźniak, Paulina Cieślik, Katarzyna Kieć-Kononowicz, Jadwiga Handzlik, Andrzej J. Bojarski
, Med. Chem. Commun.
, 2018
, 9
, 1882
- Halogen bonding enhances activity in a series of dual 5-HT6/D2 ligands designed in a hybrid bioisostere generation/virtual screening protocol. Jakub Staroń, Dawid Warszycki, Rafał Kurczab, Grzegorz Satała, Ryszard Bugno, Adam Hogendorf, Andrzej J. Bojarski
, RSC Adv.
, 2016
, 6
, 54918