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2Gil et al..
Coupling of Receptor Conformation and Ligand Orientation Determine Graded Activity, Nature Chemical Biology, 2010 Srinivasan et al.
Ligand-binding dynamics rewire cellular signaling via estrogen receptor-alpha.
Nature Chemical Biology, doi: 10.1038/nchembio.1214, published online 24 March 2013
http://www.nature.com/naturechemicalbiology, Nature Chemical Biology