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4Di Paolo et al..
Specific Btk inhibition suppresses B-cell and myeloid-cell mediated arthritis, Nature Chemical Biology, 2010 Chen Haiyang, Song Peiran, Diao Yanyan, Hao Yongjia, Dou Dou, Wang Wanqi, Fang Xiaoyu, Wang Yanling, Zhao Zhenjiang, Ding Jian, Li Honglin, Xie Hua, Xu Yufang.
Discovery and biological evaluation of N5-substituted 6,7-dioxo-6,7-dihydropteridine derivatives as potent Bruton's tyrosine kinase inhibitors, MedChemComm, 2018