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2Yoneyama, Hiroki; Magata, Takuji; Uemura, Kenji; Usami, Yoshihide; Tanaka, Satoshi; Takaoka, Masanori; Harusawa, Shinya, Synthesis 2015, 47, 1291-1302.
Efficient Synthesis of N-[4-(4-Chlorophenyl)butyl]-S-(3-piperidinopropyl)isothiourea (OUP-186) and Its Analogues Using 2-Nitrophenylacetyl Isothiocyanate: Application to Novel Histamine H3R Antagonists, Synthesis