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2Apsel et al..
Targeted polypharmacology: discovery of dual inhibitors of tyrosine and phosphoinositide kinases, Nature Chemical Biology, 2008 Bergamini et al.
A selective inhibitor reveals PI3Kgamma dependence of TH17 cell differentiation.
Nature Chemical Biology, doi: 10.1038/nchembio.957, published online 29 April 2012
http://www.nature.com/naturechemicalbiology, Nature Chemical Biology